KIT

ENSG00000157404 - H. sapiens

Pathways

Go term Description
GO:0002020 protease binding
GO:0004713 protein tyrosine kinase activity
GO:0004714 transmembrane receptor protein tyrosine kinase activity
GO:0004716 signal transducer, downstream of receptor, with protein tyrosine kinase activity
GO:0005020 stem cell factor receptor activity
GO:0005088 Ras guanyl-nucleotide exchange factor activity
GO:0005515 protein binding
GO:0005524 ATP binding
GO:0019955 cytokine binding
GO:0042803 protein homodimerization activity
GO:0046872 metal ion binding
GO:0046934 phosphatidylinositol-4,5-bisphosphate 3-kinase activity

Drugs

Drug name Description
CABOZANTINIB
DASATINIB Tyrosine-protein kinase ABL inhibitor
IMATINIB Tyrosine-protein kinase ABL inhibitor
LENVATINIB
PAZOPANIB Tyrosine-protein kinase LCK inhibitor
PONATINIB Tyrosine-protein kinase ABL inhibitor
REGORAFENIB Tyrosine-protein kinase ABL inhibitor
SORAFENIB Serine/threonine-protein kinase RAF inhibitor
SUNITINIB Macrophage colony stimulating factor receptor inhibitor

Diseases

Disease Name
GIST
AML
TGCT
mastocytosis
mucosal melanoma
epithelioma

Orthologs

Gene Organism
Pvr D. melanogaster

Related Interactions

Gene ID A Gene Name A Gene ID B Gene Symbol B Organism Source Score?
ENSG00000072274 TFRC ENSG00000157404 KIT H. sapiens SSL Slorth 0.786913 View
ENSG00000100644 HIF1A ENSG00000157404 KIT H. sapiens SSL Slorth 0.786826 View
ENSG00000112658 SRF ENSG00000157404 KIT H. sapiens SSL Slorth 0.786236 View
ENSG00000101199 ARFGAP1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.785949 View
ENSG00000132906 CASP9 ENSG00000157404 KIT H. sapiens SSL Slorth 0.785835 View
ENSG00000063244 U2AF2 ENSG00000157404 KIT H. sapiens SSL Slorth 0.78583 View
ENSG00000074181 NOTCH3 ENSG00000157404 KIT H. sapiens SSL Slorth 0.784627 View
ENSG00000136527 TRA2B ENSG00000157404 KIT H. sapiens SSL Slorth 0.784219 View
ENSG00000101557 USP14 ENSG00000157404 KIT H. sapiens SSL Slorth 0.783931 View
ENSG00000094916 CBX5 ENSG00000157404 KIT H. sapiens SSL Slorth 0.783199 View
ENSG00000157404 KIT ENSG00000166167 BTRC H. sapiens SSL Slorth 0.783009 View
ENSG00000118640 VAMP8 ENSG00000157404 KIT H. sapiens SSL Slorth 0.782734 View
ENSG00000138696 BMPR1B ENSG00000157404 KIT H. sapiens SSL Slorth 0.782719 View
ENSG00000005007 UPF1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.782661 View
ENSG00000157404 KIT ENSG00000185651 UBE2L3 H. sapiens SSL Slorth 0.782571 View
ENSG00000066654 THUMPD1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.782557 View
ENSG00000007168 PAFAH1B1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.782524 View
ENSG00000157404 KIT ENSG00000185359 HGS H. sapiens SSL Slorth 0.78227 View
ENSG00000157404 KIT ENSG00000166508 MCM7 H. sapiens SSL Slorth 0.781974 View
ENSG00000119318 RAD23B ENSG00000157404 KIT H. sapiens SSL Slorth 0.781786 View
ENSG00000123159 GIPC1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.78162 View
ENSG00000135521 LTV1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.78067 View
ENSG00000157404 KIT ENSG00000245848 CEBPA H. sapiens SSL Slorth 0.780663 View
ENSG00000119912 IDE ENSG00000157404 KIT H. sapiens SSL Slorth 0.780572 View
ENSG00000108561 C1QBP ENSG00000157404 KIT H. sapiens SSL Slorth 0.78009 View
ENSG00000153107 ANAPC1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.779306 View
ENSG00000117758 STX12 ENSG00000157404 KIT H. sapiens SSL Slorth 0.779304 View
ENSG00000064012 CASP8 ENSG00000157404 KIT H. sapiens SSL Slorth 0.779288 View
ENSG00000004487 KDM1A ENSG00000157404 KIT H. sapiens SSL Slorth 0.778992 View
ENSG00000116350 SRSF4 ENSG00000157404 KIT H. sapiens SSL Slorth 0.778361 View
ENSG00000113812 ACTR8 ENSG00000157404 KIT H. sapiens SSL Slorth 0.777739 View
ENSG00000075413 MARK3 ENSG00000157404 KIT H. sapiens SSL Slorth 0.777243 View
ENSG00000157404 KIT ENSG00000170606 HSPA4 H. sapiens SSL Slorth 0.776885 View
ENSG00000157404 KIT ENSG00000188021 UBQLN2 H. sapiens SSL Slorth 0.776611 View
ENSG00000157404 KIT ENSG00000185345 PARK2 H. sapiens SSL Slorth 0.77631 View
ENSG00000130811 EIF3G ENSG00000157404 KIT H. sapiens SSL Slorth 0.776147 View
ENSG00000113722 CDX1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.776106 View
ENSG00000156304 SCAF4 ENSG00000157404 KIT H. sapiens SSL Slorth 0.775881 View
ENSG00000079102 RUNX1T1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.775408 View
ENSG00000137815 RTF1 ENSG00000157404 KIT H. sapiens SSL Slorth 0.775023 View